Population Pharmacokinetic Evaluation of Eslicarbazepine Acetate for Adjunctive Therapy in Refractory Partial Onset Seizures

Population Pharmacokinetic Evaluation of Eslicarbazepine Acetate for Adjunctive Therapy in Refractory Partial Onset Seizures

Conference: ACCP

Eslicarbazepine acetate (ESL), a once-daily antiepileptic drug (AED), is converted to eslicarbazepine, the primary active metabolite of ESL, after oral administration. The population pharmacokinetics (PK)…

Design, Synthesis, and in vitro Testing of Novel COX-2/COX-1 Inhibitors

Design, Synthesis, and in vitro Testing of Novel COX-2/COX-1 Inhibitors

Division: PBPK

To design,synthesize,and test new lead molecules that inhibit both COX-1 and COX-2 forms of the cyclooxygenase (COX) enzyme, with higher affinity for COX-2 than for COX-1.

3D QSAR and pharmacophore study of curcuminoids and curcumin analogs: Interaction with thioredoxin reductase

3D QSAR and pharmacophore study of curcuminoids and curcumin analogs: Interaction with thioredoxin reductase

Publication: Interdiscip Sci
Software: ADMET Predictor®

Curcumin is the yellow pigment of Curcuma longa that irreversibly inhibits the activity of thioredoxin reductase (TrxR) and forms adduct.

Preoperative androgen deprivation therapy for localized prostate cancer: delayed biochemical recurrence in high-risk disease

Preoperative androgen deprivation therapy for localized prostate cancer: delayed biochemical recurrence in high-risk disease

Publication: Clin Genitourin Cancer

Background: The role of preoperative ADT for localized prostate cancer is controversial; prospective assessments have yielded varying results. We sought to define a subset...

Prediction of Valsartan Pharmacokinetics in Pediatric Population using Physiologically Based Pharmacokinetic (PBPK) Model

Prediction of Valsartan Pharmacokinetics in Pediatric Population using Physiologically Based Pharmacokinetic (PBPK) Model

Conference: AAPS
Software: GastroPlus®
Division: PBPK

A method for transporter-based in vitro-in vivo extrapolation (IVIVE) was previously developed and demonstrated by predicting valsartan PK after i.v.administration [1]. The purpose of this study was to…