Why Next-Generation Mechanistic Models will Transform Drug Discovery: Integrating Efficacy and Safety

Why Next-Generation Mechanistic Models will Transform Drug Discovery: Integrating Efficacy and Safety

Publication: Expert Opin Drug Discov
Software: DILIsym®, GastroPlus®

Drug discovery remains constrained by high attrition rates and the fragmented evaluation of exposure, efficacy, and safety.

Animal-Free Skin Sensitization Testing: In Chemico and In Silico Integrated Approach

Animal-Free Skin Sensitization Testing: In Chemico and In Silico Integrated Approach

Publication: Toxics
Software: ADMET Predictor®

The increasing prohibition of animal testing for cosmetic products has driven the development of alternative approaches to ensure consumer safety.

Sex-Related Differences in Physiologically-Based Biopharmaceutics Modeling

Sex-Related Differences in Physiologically-Based Biopharmaceutics Modeling

Publication: CPT Pharmacometrics Syst Pharmacol
Software: GastroPlus®

Physiologically based pharmacokinetic (PBPK) and physiologically-based biopharmaceutics (PBBM) modeling are valuable tools in drug development, allowing mechanistic predictions of drug absorption and disposition.

Integrated Population Pharmacokinetic and Exposure-Response Modeling of Enlicitide in Hypercholesterolemia Patients Supports Clinical Dose Recommendation Across Patient Subgroups

Integrated Population Pharmacokinetic and Exposure-Response Modeling of Enlicitide in Hypercholesterolemia Patients Supports Clinical Dose Recommendation Across Patient Subgroups

Conference: PAGE

Despite the well-established cardiovascular benefit of  low-density lipoprotein cholesterol (LDL-C) lowering, real-world use of  PCSK9-targeted therapies remains limited, in part due to reliance on injectable formulations.

2025 AAPS 360 Annual Meeting: Highlights in In Vitro Release and Dissolution Testing and Oral Biopharmaceutics Modeling

2025 AAPS 360 Annual Meeting: Highlights in In Vitro Release and Dissolution Testing and Oral Biopharmaceutics Modeling

Publication: Dissolution Tech
Software: GastroPlus®

This manuscript highlights key sessions from the In Vitro Release and Dissolution Testing (IVRDT) and Oral Biopharmaceutics and Absorption Modeling (OBAM) communities at the 2025 AAPS PharmSci 360 Annual Meeting (November 9–12, San Antonio, TX).

Impact of Preclinical Verification in Physiologically Based Pharmacokinetic Modelling for First-in-Human Predictions: Application of a Published Model Building Strategy for Five Compounds

Impact of Preclinical Verification in Physiologically Based Pharmacokinetic Modelling for First-in-Human Predictions: Application of a Published Model Building Strategy for Five Compounds

Publication: Clinical Pharmacokinetics
Software: GastroPlus®

Physiologically based pharmacokinetic modelling is routinely used in the pharmaceutical industry and has an impact on drug labels.