In Silico Predictions for ADME and Toxicology

In Silico Predictions for ADME and Toxicology

Publication: CRC Press
Software: ADMET Predictor®

Advances in computational modeling are transforming how scientists predict a compound’s Absorption, Distribution, Metabolism, Excretion, and Toxicology (ADMET) profiles.

In Silico Prediction of Solubility, Permeability, and Metabolism

In Silico Prediction of Solubility, Permeability, and Metabolism

Publication: CRC Press

This chapter presents a comprehensive review of in silico techniques for the prediction of solubility, permeability, and metabolism—critical determinants of drug candidates’ pharmacokinetic and safety profiles during drug discovery and development.

Physiologically Based Pharmacokinetic Modeling of Cefotaxime To Inform Pediatric Dosing in Renal Impairment

Physiologically Based Pharmacokinetic Modeling of Cefotaxime To Inform Pediatric Dosing in Renal Impairment

Publication: Eur J Clin Pharmacol
Software: GastroPlus®

Cefotaxime (CFT) is a broad spectrum, third-generation cephalosporin antibiotic prescribed for the treatment of severe infections, yet dosing guidelines for pediatric with renal impairment is scarce.

Why Next-Generation Mechanistic Models will Transform Drug Discovery: Integrating Efficacy and Safety

Why Next-Generation Mechanistic Models will Transform Drug Discovery: Integrating Efficacy and Safety

Publication: Expert Opin Drug Discov
Software: DILIsym®, GastroPlus®

Drug discovery remains constrained by high attrition rates and the fragmented evaluation of exposure, efficacy, and safety.

Animal-Free Skin Sensitization Testing: In Chemico and In Silico Integrated Approach

Animal-Free Skin Sensitization Testing: In Chemico and In Silico Integrated Approach

Publication: Toxics
Software: ADMET Predictor®

The increasing prohibition of animal testing for cosmetic products has driven the development of alternative approaches to ensure consumer safety.

2025 AAPS 360 Annual Meeting: Highlights in In Vitro Release and Dissolution Testing and Oral Biopharmaceutics Modeling

2025 AAPS 360 Annual Meeting: Highlights in In Vitro Release and Dissolution Testing and Oral Biopharmaceutics Modeling

Publication: Dissolution Tech
Software: GastroPlus®

This manuscript highlights key sessions from the In Vitro Release and Dissolution Testing (IVRDT) and Oral Biopharmaceutics and Absorption Modeling (OBAM) communities at the 2025 AAPS PharmSci 360 Annual Meeting (November 9–12, San Antonio, TX).